Tag: bet

Pharma / Biotech

Novel phenanthridin-6(5H)-one derivatives as potent and selective BET bromodomain inhibitors: Rational design, synthesis and biological evaluation.

Newsemia
Related Articles Novel phenanthridin-6(5H)-one derivatives as potent and selective BET bromodomain inhibitors: Rational design, synthesis and biological evaluation. Eur J Med Chem. 2019 Jun 28;179:502-514...
Pharma / Biotech

Exploiting the 7-methylimidazo[1,5-a]pyrazin-8(7H)-one scaffold for the development of novel chemical inhibitors for Bromodomain and Extraterminal Domain (BET) family.

Newsemia
Related Articles Exploiting the 7-methylimidazo[1,5-a]pyrazin-8(7H)-one scaffold for the development of novel chemical inhibitors for Bromodomain and Extraterminal Domain (BET) family. Bioorg Chem. 2019 Jun 11;90:103044...
Pharma / Biotech

Characterizing the Therapeutic Potential of a Potent BET Degrader in Merkel Cell Carcinoma.

Newsemia
Related Articles Characterizing the Therapeutic Potential of a Potent BET Degrader in Merkel Cell Carcinoma. Neoplasia. 2019 Feb 20;21(3):322-330 Authors: Choi JE, Verhaegen ME, Yazdani...

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